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美国ActiveBiochem公司产品价格目录

美国ActiveBiochem公司产品价格目录

美国ActiveBiochem公司产品价格目录

蚂蚁淘(ebiomall)是一家生命科学领域的垂直电商平台,公司专注生物医学科研用品的  全球导购和品牌推广,为海外厂方与国内代理经销商搭建跨境贸易系统和交流平台。

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借助互联网平等而开放的力量,矢志实现生命科学领域全球的信息同步,我们相信一群充满梦想的人,可以凭借着专业与执着,让你的购物更轻松!

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关于美国ActiveBiochem公司

ActiveBiochem是小分子抗癌剂,激酶抑制剂和其他生物活性剂的领先供应商。我们承诺以具有竞争力的价格提供最好的质量。
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美国ActiveBiochem公司产品价格目录


MIK-665(S-64315)(Catalog#:A-1457)(Target:MCL-1)(CAS#:1799631-75-6)MIK-665(S-64315)isaninhibitorofinducedmyeloidleukemiacelldifferentiationprotein(Mcl-1;B...Rocaglamide(Catalog#:A-1624)(Target:NF-κB)(CAS#:84573-16-0)Rocaglamideisanimmunosuppressant,andapotentinhibitorofNF-κBactivationinTcells,withan...E-7090(Catalog#:A-6063)(Target:FGFR)(CAS#:1622204-21-0)E-7090isaselectiveinhibitorofthetyrosinekinaseactivitiesofFGFR1,-2,and-3....CB-1158(Catalog#:A-6098)(Target:Arginase)(CAS#:2095732-06-0)CB-1158isapotentinhibitorofhumanarginase(IC50=98nM).Inculture,humangranulocytesrelea...BAY-1816032(Catalog#:A-1166)(Target:BUB1)(CAS#:1891087-61-8)BAY-1816032isapotentandselectiveBUB1(Mitoticcheckpointserine/threonine-proteinkinase)inhi...IPI-926(Saridegib)(Catalog#:A-1062)(Target:Hedgehog)(CAS#:1037210-93-7)IPI-926(Saridegib)isanorallybioavailableinhibitoroftheHedgehog(Hh)pathwaywithpotential...BLU-285(Avapritinib)(Catalog#:A-1222)(Target:KIT;PDGFRα)(CAS#:1703793-34-3)BLU-285isapotentandselectiveinhibitorofPDGFRα(D842V)andKITExon17mutants....PD-1/PDL-1Inhibitor1(Catalog#:A-9111)(Target:PD-1/PDL-1Interaction)(CAS#:1675201-83-8 )PD-1/PD-L1inhibitor1isasmall-moleculeinhibitorofPD-1/PD-L1interactionatIC50of6nM....S-63845(Catalog#:A-6044)(Target:MCL-1)(CAS#:1799633-27-4 )S-63845isapotentandselectiveMCL1inhibitor(Ki(MCL1,FP)<1.2nM;Kd(MCL1,SPR)=0.19nM;...FF-10101(Catalog#:A-9114)(Target:FLT3)(CAS#:1472797-69-5(freebase))FF-10101isanovelirreversIBLeFLT3inhibitor,andshowsexcellentefficacyagainstAMLcellswith...(+)-EtomoxirSodiumSaltHydrate(Catalog#:A-1672)(Target:CPT1)(CAS#:828934-41-4)...ARS-1620(Catalog#:A-1671)(Target:K-RAS(G12C))(CAS#:1698055-85-4)ARS-1620isapotentandirreversibleinhibitorofmutantK-RAS(G12C)throughacovalentbondwitht...THZ-531(Catalog#:A-1670)(Target:CDK12;CDK13)(CAS#:1702809-17-3)...EPZ-031686(Catalog#:A-1669)(Target:SMYD3;MEKK2)(CAS#:1808011-22-4)EPZ-031686isanoncompetitiveinhibitorforSMYD3andMEKK2withaKi=1.2and1.1nMrespectively....eFT-226(Catalog#:A-1668)(Target:eIF4A)(CAS#:)eFT-226isaselectiveandhighlypotentinhibitorofeukaryoticinitiationfactor4A(eIF4A),anov...SEL120-34A(Catalog#:A-2554)(Target:CDK8)(CAS#:1609452-30-3(HCl))SEL120-34AisapotentandselectiveCDK8inhibitoractiveinAMLcellswithhighlevelsofserinep...MK-0731(Catalog#:A-1298)(Target:KSP)(CAS#:845256-65-7)MK-0731isapotentandselectiveinhibitorofkinesinspindleprotein(KSP),whichmayresultinth...RDEA-436(Catalog#:A-1038)(Target:)(CAS#:)RDEA-436isasecond-generationmitogen-activatedERKkinaseinhibitorforthetreatmentofcancer....PT-2385(Catalog#:A-1510)(Target:HIF)(CAS#:1672665-49-4)PT-2385isanorallyactive,smallmoleculeinhibitorofhypoxiainduciblefactor(HIF)-2alpha,with...ASTX-660(Catalog#:A-9109)(Target:XIAP,cIAP1)(CAS#:1799328-86-1)ASTX-660isanorallybioavailable,non-peptidomimeticantagoNISTofbothXchromosome-linkedinhibi...AZD-1390(Catalog#:A-9108)(Target:ATM)(CAS#:2089288-03-7)AZD1390isapotentandselectiveATMinhibitor....BAY-1143572(Catalog#:A-1514)(Target:CDK)(CAS#:)BAY-1143572isahighlyselective,potentandorallyavailableinhibitorofPTEFb/CDK9.BAY-1143572...BMS-906024(Catalog#:A-1401)(Target:Notch)(CAS#:1401066-79-2)BMS-906024isapotentandselectiveNotchreceptorinhibitor....FGF-401(Catalog#:A-6073)(Target:FGFR4)(CAS#:1708971-55-4)FGF-401isaninhibitorofhumanfibroblastgrowthfactorreceptor4(FGFR4),withpotentialantineo...BMS-986205(Catalog#:A-6067)(Target:IDO1)(CAS#:1923833-60-6)BMS-986205isanoptimized,potent,selectiveandorallybioavailableIDO1(indoleamine2,3-dioxygen...GSK-2194069(Catalog#:A-6000)(Target:hFAS)(CAS#:1332331-08-4 )GSK-2194069isapotentandselectivehumanfattyacidsynthase(hFAS)inhibitor(IC50=7.7nM).Hu...GSK-126(Catalog#:A-1275)(Target:EZH2)(CAS#:1346574-57-9)GSK-126isapotent,highlyselective,S-adenosyl-methionine-competitive,small-moleculeinhibitoro...ASP-2215(Gilteritinib)(Catalog#:A-1371)(Target:FLT3;AXL)(CAS#:1254053-43-4)ASP-2215(Gilteritinib)isapotentFLT3/AXLinhibitor,showingstronganti-leukemicactivityagains...ARQ-087(Derazantinib)(Catalog#:A-6001)(Target:FGFR)(CAS#:1234356-69-4)ARQ-087(Derazantinib)isanorallybioavailableinhibitorofthefibroblastgrowthfactorreceptor...EED-226(Catalog#:A-9102)(Target:EZH2)(CAS#:2083627-02-3)EED-226isafirst-in-classpotent,selective,andorallybioavailableEED(EmbryonicEctodermDevel...LY-3009120(DP-4978)(Catalog#:A-1317)(Target:RAF)(CAS#:1454682-72-4)LY-3009120(DP-4978)ispotentandselectivepan-RAFinhibitorwithpotentialanticanceractivity.L...E-7046(Catalog#:A-1336)(Target:PGE2)(CAS#:1369489-71-3)E-7046isaspecificantagonistofthetype4prostaglandinE2(PGE2)receptorEP4.Itpossessessig...PQR-530(Catalog#:A-1479)(Target:PI3K;mTOR )(CAS#:1927857-61-1)PQR-530isapanPI3K/mTORInhibitor....AG-881(Vorasidenib)(Catalog#:A-6078)(Target:IDH1,IDH2 )(CAS#:1644545-52-7)AG-881(Vorasidenib)isapotentandselectiveorallyavailableinhibitorofmutatedformsofbothi...CFI-400945(FreeBase)(Catalog#:A-6005)(Target:PLK4)(CAS#:1338806-73-7)CFI-400945isanorallyavailablePLK4(polo-likekinase4)inhibitorwithpotentialantineoplastic...CPI-444(Catalog#:A-6099)(Target:A2A)(CAS#:1202402-40-1)CPI-444isasmallmoleculeimmunecheckpointinhibitoroftheadenosineA2Areceptor(ADORA2A)with...TPX-0005(Catalog#:A-1507)(Target:ALK;ROS1;TRK)(CAS#:1802220-02-5)TPX-0005isapotentALK/ROS1/TRKinhibitor.TPX-0005effectivelyinhibitedabroadspectrumofmuta...FT-1518(Catalog#:A-1419)(Target:mTOR)(CAS#:1313026-58-2)FT-1518isapotentandselectivemTORInhibitor....ON-123300(Catalog#:A-1465)(Target:ARK5;CDK4)(CAS#:1357470-29-1 )ON-123300isapotentmultikinaseinhibitorofARK5andCDK4,aswellasgrowthfactorreceptortyro...MTX-211(Catalog#:A-1462)(Target:PI3K;EGFR)(CAS#:1952236-05-3)MTX-211isafirst-in-classdualinhibitorofPI3KandEGFRkinaseswithdemonstratedinvivoantica...NVP-CGM-097(CGM-097)(Catalog#:A-1464)(Target:MDM2)(CAS#:1313363-54-0)NVP-CGM-097(CGM-097)isanorallybioavailableHDM2(humanhomologofdoubleminute2)antagonistw...BLU-554(Catalog#:A-6071)(Target:FGFR4)(CAS#:1707289-21-1)BLU-554isapotent,orallybioavailableinhibitorofhumanfibroblastgrowthfactorreceptor4(FGF...GDC-0084(Catalog#:A-6015)(Target:PI3K)(CAS#:1382979-44-3)GDC-0084isapotentPI3Kinhibitorwithantineoplasticactivity.GDC-0084specificallyinhibitsPI3...AvitinibMaleate(Catalog#:A-6109)(Target:EGFR)(CAS#:1557268-88-8(maleate) )Avitinib(AC0010,AC0010MA)isanorallyavailable,irreversible,epidermalgrowthfactorreceptor(...BGB-324(R-428)(Catalog#:A-6103)(Target:AXL)(CAS#:1037624-75-1 )BGB-324(R-428)isaselectiveandpotentinhibitorofAXLkinase,whichshowedactivitytoblockst...LXS-196(Catalog#:A-6075)(Target:PKC)(CAS#:1874276-76-2)LXS-196isanorallyavailableproteinkinaseC(PKC)inhibitorwithpotentialimmunosuppressiveand...H3B-6527(Catalog#:A-6107)(Target:FGFR4)(CAS#:1702259-66-2 )H3B-6527isapotent,selectiveandorallybioavailableinhibitorofhumanFGFR4(fibroblastgrowth...BGB-290(Catalog#:A-6108)(Target:PARP)(CAS#:1446261-44-4)BGB-290isapotentandorallybioavailableinhibitorofthenuclearenzymepoly(ADP-ribose)polymer...BAY-1082439(Catalog#:A-6042)(Target:PI3Kα/β)(CAS#:1375469-38-7 )BAY-1082439isanorallybioavailableinhibitoroftheclassIphosphoinositide3-kinase(PI3K)alph...ABL-001(Asciminib)(Catalog#:A-1967)(Target:BCR-ABL)(CAS#:1492952-76-7)ABL-001(Asciminib)isapotentallostericinhibitorofBCR-ABL.ABL001preventsemergenceofresist...BLU-9931(Catalog#:A-1397)(Target:FGFR4)(CAS#:1538604-68-0)BLU-9931isapotentandirreversiblesmall-moleculeinhibitorofFGFR4.BLU-9931isexquisitelyse...BAY-876(Catalog#:A-6009)(Target:GLUT1)(CAS#:1799753-84-6)BAY-876isapotentandselectiveGLUT1Inhibitor,withgoodmetabolicstABIlityin vitroandhigh...MI-503(Catalog#:A-1399)(Target:Menin-MLLinteraction)(CAS#:1857417-13-0)MI-503isahighlypotentandorallybioavailablesmallmoleculeinhibitorofthemenin-MLLinteract...

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