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商品描述
B-Raf IN 1
- Catalog No.:MC0629
- Data Sheet
- MSDS
- Support
- Description
- References ( 0 )
- Protocol
- CasNo:
- 950736-05-7
- MolecularFormula:
- C29H24F3N5O
- Purity:
- >98%
- Target:
- Raf
- IC50:
- No data
- Fields:
- B-Raf IN 1 is a highlt potent and selective B-Raf inhibitor with IC50 of 24 nM; equipotent against c-Raf (IC50= 25 nM).
- Specificity:
- Target: Raf . Fields: B-Raf IN 1 is a highlt potent and selective B-Raf inhibitor with IC50 of 24 nM; equipotent against c-Raf (IC50= 25 nM).
- Source:
- Rabbit
- Dilution:
- WB 1:500-2000
- Concentration:
- >98%
- Storage Stability:
- 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
- MolecularWeight(Da):
- 515.53
- References:
- [1]. Berger DM, et al. Non-hinge-binding pyrazolo[1,5-a]pyrimidines as potent B-Raf kinase inhibitors. Bioorg Med Chem Lett. 2009 Dec 1;19(23):6519-23.
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