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0512-67156496
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商品描述
ACY-738
- Catalog No.:MC0952
- Data Sheet
- MSDS
- Support
- Description
- References ( 0 )
- Protocol
- CasNo:
- 1375465-91-0
- MolecularFormula:
- C14H14N4O2
- Purity:
- >98%
- Target:
- HDAC
- IC50:
- No data
- Fields:
- ACY-738 demonstrates inhibitory activity against recombinant HDAC6 with IC50 values of 1.7 nM, with respective average selectivity over class I HDACs being 100-fold.
- Specificity:
- Target: HDAC . Fields: ACY-738 demonstrates inhibitory activity against recombinant HDAC6 with IC50 values of 1.7 nM, with respective average selectivity over class I HDACs being 100-fold.
- Source:
- Rabbit
- Dilution:
- WB 1:500-2000
- Concentration:
- >98%
- Storage Stability:
- 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
- Other Name:
- ACY738,ACY-738,ACY 738
- MolecularWeight(Da):
- 270.29
- References:
- [1]. Jochems J, et al. Antidepressant-like properties of novel HDAC6-selective inhibitors with improved brain bioavailability. Neuropsychopharmacology. 2014 Jan;39(2):389-400.
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