Description | SGC-GAK-1isapotent,selective,andcell-activeinhibitorofcyclinG-associatedkinase(GAK)withKivalueof3.1nMand>50-foldselectivityovernearestkinase. | ||
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Targets |
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Invitro | SGC-GAK-1showsstronggrowthinhibitioninLNCaP,VCaP,and22Rv1cellsat10μM,butminimaleffectinPC3andDU145cells.IndoseresponseSGC-GAK-1showspotentantiproliferativeactivityinLNCaPand22Rv1cellsatasimilardoserangethatitengagesGAK[1]. |