FormuMax/Alendrosome™ - Alendronate Liposomes (Neutral)/F70103A-N/

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¥11980.00
货号:F70103A-N
浏览量:127
品牌:FormuMax
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商品描述

Alendrosome™-Alendronateliposomes(Neutral)

WearelookingforresearcherstotestourAlendrosome™products,pleasecontactusifyouareinterested

Specifications

Active:alendronatesodium(CAS121268-17-5),2.0mg/mL

Alendronate Sodium

Volume:10.0mL

Lipidcomposition:phosphatidylcholineandcholesterol

Internal/Externalsolution:phosphatebufferedsaline(20mMsodiumphosphate,09wt%NaCl),pH7.0-7.5

Usage:warmtoroomtemperatureandmixwellbeforeuse.

Dosage:thisisanewproductandnorecommendeddoseisavailableatthispoint.Referthefollowingliteratureforadditionalinformation

References

BenjaminJ.Burwitzetal.TechnicalAdvance:Liposomalalendronatedepletesmonocytesandmacrophagesinthenonhumanprimatemodelofhumandisease.JLeukocBiol.2014Sep;96(3):491–501.PMC4632165(Link)

RenateFrei,Comparisonofcytotoxicpropertiesoffreeandliposomalbisphosphonatesinvitro(DiplomaThesis)(Link)

MönkkönenJ,vanRooijenN,YlitaloP.,EffectsofClodronateandpamidronateonsplenicandhepaticphagocyticcellsofmice.PharmacolToxicol.1991Apr;68(4):284-6.(Link)
MakkonenN,HirvonenMR,TeräväinenT,SavolainenK,MönkkönenJ.,DifferenteffectsofthreebisphosphonatesonnitricoxideproductionbyRAW264macrophage-likecellsinvitro.JPharmacolExpTher.1996May;277(2):1097-102(link)
vanRooijenN,KorsN.Effectsofintracellulardiphosphonatesoncellsofthemononuclearphagocytesystem:invivoeffectsofliposome-encapsulateddiphosphonatesondifferentmacrophagesubpopulationsinthespleen.CalcifTissueInt.1989Sep;45(3):153-6.(Link)
EpsteinH.etal.,PreparationofalendronateliposomesforenhancedstABIlityandbioactivity:invitroandinvivocharacterization.AAPSJ.2008Dec;10(4):505-15.Epub2008Oct21.(Link)
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