TM-2-51Highly potentand isozyme selective activator of recombinant HDAC8. Increases the activity of HDAC8 by a factor of12 at 10 µM.No activation of other HDACs is observed. Rescues the activity of catalyticallycompromised HDAC8 mutants in vitro.Amount:10mgPhysical Properties:BeigepowderMW=256.3 C14H12N2OS
Analysis:>98%(TLC); NMR (Conforms)
Solubilization:May be dissolved in DMSO (50 mg/ml); or ethanol (8 mg/ml)
Storage:Storedesiccated as supplied at -20°C for up to 2 years. Store solutions at-20°C for up to 3 months.
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