CI-994 N-acetyldinaline;4-(Acetylamino)-N-(2-aminophenyl)benzamide; PD-123654
CI-994 is an orally active histone deacetylase (HDAC) inhibitor, IC50 = 0.9,0.9, 1.2 and >20 µM for HDAC1, HDAC2, HDAC3 and HDAC8 respectively.Mediates G1 cell cycle arrest, inhibits proliferation and inducesapoptosis in vitro and in vivo. Increaseneuroplasticity during memory extinction. Protects beta cells fromcytokine-induced apoptosis.
Physical Properties: Off-white powder
MW=269.3 C15H15N3O2
Analysis: >98% (TLC); NMR(Conforms)
Solubilization: May be dissolved in DMSO (25 mg/ml)
Storage: Store desiccated assupplied at -20°C for up to 2 years. Store solutions at -20°C for up to 1 month.
Amount: 5mg
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