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联系方式
公司地址
苏州工业园区生物纳米园A4#216
联系电话
4000-520-616 / 18915418616
传真号码
0512-67156496
电子邮箱
info@ebiomall.com
公司网址
https://www.ebiomall.com
商品描述
- VerypotentEGFreceptorkinase(tyrosinekinase)inhibitor(IC50=3nM).VeryweakonPDGFreceptorandHER2-NEUkinases(IC50>100µM).Osherov,N.andLevitzki,A."Epidermal-growth-factor-dependentactivationofthesrc-familykinases."Eur.J.Biochem.225:1047-1053(1994).Levitzki,A.andGazit,A."Tyrosinekinaseinhibition:anapproachtodrugdevelopment."Science267:1782-1788(1995).
- ReversIBLyinhibits(IC50=9.8µM)theratbrainKv1.5potassiumchannelinvitroinanon-protein-tyrosine-kinase-mediatedmanner.Choi,B.H.,etal."DirectinhibitionoftheclonedKv1.5channelbyAG-1478,atyrosinekinaseinhibitor."Am.J.Physiol.CellPhysiol.282:C1461-C1468(2002).
- Soldforlaboratoryormanufacturingpurposesonly;notforhuman,medical,veterinary,food,orhouseholduse.
RelatedTerms:
[AG1478]M.W.315.75
C16H14ClN3O2
[175178-82-2]